
UFR : Pharmacie Clermont-Ferrand
Nom : COUDERT
Prénom : Pascal
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Equipe de recherche
- Intitulé : Imagerie Moléculaire et Thérapie Vectorisée
- Numéro : 990
- Thématiques : Vectorisation de principes actifs à activité antitumorale
Mots clés : chlorambucil, fluoro-uracil, fluorodeoxyglucose, antitumour activity
Principales publications
- Synthesis and cytotoxic properties of new fluorodeoxyglucose-coupled chlorambucil derivatives, B. REUX, V. WEBER, M-J GALMIER, M. BOREL, M. MADESCLAIRE, J-C. MADELMONT, E. DEBITON and P. COUDERT, Bioorg. Med. Chem., 2008, 16, 5004-5020.
- Preclinical investigation of tolerance and antitumour activity of new fluorodeoxyglucose-coupled chlorambucil alkylating agents, E. MIOT-NOIRAULT, B. REUX, E. DEBITON, J-C. MADELMONT, J-M. CHEZAL, P. COUDERT and V. WEBER, Invest. New Drugs, 2011, 29, 424-433.
- Design, synthesis and in vitro drug release investigation of new potential 5-FU prodrugs, P. DAUMAR, C. DECOMBAT, J-M CHEZAL, E. DEBITON, M. MADESCLAIRE, P. COUDERT and M-J GALMIER, Eur. J. Med. Chem., 2011, 46, 2867-2879.
- Reactions of (S)-(4-nitrophenyl)[(4S)-2-oxo-1,3-oxazolidin-4yl]methyl methanesulfonate with alkali metal halides and lithium hydroxide. Synthesis of [(2R, 3R)-3-(4-nitrophenyl)aziridin-2-yl] methanol, M. MADESCLAIRE, P. COUDERT, F. LEAL, S. TARRIT, YU. V. ZAITSEVA and V. P. ZAITSEV, Chem. Het. Comp., 2013, 49, 1103-1107.
- Synthesis and antimicrobial activity of new ureas from (1S,2S)-2-amino-1-(4-nitrophenyl)-1,3-propanediol. M. MADESCLAIRE, P. COUDERT, A.V. LYAMIN, S. Kh. SHARIPOVA, YU. V. ZAITSEVA and V. P. ZAITSEV, Pharmaceutical Chemistry Journal, 2015, 49, n°1, 10-12.




